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BTK

Brief Information

Name:Tyrosine-protein kinase BTK
Target Synonym:EC 2.7.10,Bruton S Tyrosine Kinase,IGHD3,EC:2.7.10.2,Tyrosine-protein kinase BTK,AGMX1,ATK,BTK,Bruton Tyrosine Kinase,Bruton Agammaglobulinemia Tyrosine Kinase,B-Cell Progenitor Kinase,Brutons Tyrosine Kinase,BPK,Tyrosine-Protein Kinase BTK Isoform (Lacking Exon 13 To 17),Dominant-Negative Kinase-Deficient Brutons Tyrosine Kinase,Tyrosine-Protein Kinase BTK Isoform (Lacking Exon 14),Truncated Bruton Agammaglobulinemia Tyrosine Kinase,Agammaglobulinaemia Tyrosine Kinase,Agammaglobulinemia Tyrosin
Number of Launched Drugs:6
Number of Drugs in Clinical Trials:64
Lastest Research Phase:Approved

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Cat. No. Species Product Description Structure Purity Feature
BTK-H55H3 Human Human BTK Protein, His Tag (active enzyme)
BTK-H55H3-structure
BTK-H55H3-sds
ACRO Quality

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Orelabrutinib ICP-022; BIIB-135 Approved Beijing Innocare Pharma Tech Co Ltd 宜诺凯, INNOBRUKA, YINUOKAI Mainland China Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell Beijing Innocare Pharma Tech Co Ltd 2020-12-25 Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell; Central Nervous System Lymphoma; Waldenstrom Macroglobulinemia; Lymphoma; Hepatic Insufficiency; Leukemia, B-Cell; Neuromyelitis Optica; Lupus Erythematosus, Systemic; Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis; Lymphoma, Large B-Cell, Diffuse; Arthritis, Rheumatoid; Helicobacter pylori infection; Lymphoma, B-Cell, Marginal Zone; Purpura, Thrombocytopenic, Idiopathic; Lymphoma, B-Cell Details
Ibrutinib PCI-32765; CRA-032765; JNJ-54179060; PCI-32765-00 Approved Pharmacyclics Llc Imbruvica, 亿珂 United States Leukemia, Lymphocytic, Chronic, B-Cell Pharmacyclics Inc 2013-11-13 Waldenstrom Macroglobulinemia; Monoclonal Gammopathy of Undetermined Significance; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Food Hypersensitivity; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Anemia, Aplastic; Prostatic Neoplasms; Leukemia, Prolymphocytic, B-Cell; Hepatic Insufficiency; Leukemia, B-Cell; Lymphoproliferative Disorders; Leukemia, Mast-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Neoplasms, Gonadal Tissue; Intraocular Lymphoma; Lung Neoplasms; Leukemia, Myeloid, Acute; Burkitt Lymphoma; Lymphoma, T-Cell; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell; Melanoma; Leukemia, Biphenotypic, Acute; Hepatitis B, Chronic; Leukemia; Skin Melanoma; Lymphoma, B-Cell, Marginal Zone; Immunoproliferative Small Intestinal Disease; Hematopoietic stem cell transplantation (HSCT); Leukemia, Myelogenous, Chronic; HIV Infections; Hematologic Neoplasms; Solid tumours; Carcinoid Tumor; Leukemia, Lymphoid; Esophageal Neoplasms; Lymphoma, B-Cell Details
Acalabrutinib ACP-196 Approved Astrazeneca Plc, Acerta Pharma Llc Calquence, 康可期 United States Lymphoma, Mantle-Cell Astrazeneca Plc 2017-10-31 Multiple Myeloma; Leukemia, Prolymphocytic; Carcinoma, Non-Small-Cell Lung; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell; Burkitt Lymphoma; Waldenstrom Macroglobulinemia; Lymphoma; Lymphoma, Non-Hodgkin; Hepatic Insufficiency; Precursor B-Cell Lymphoblastic Leukemia-Lymphoma; Lymphoma, Follicular; Food Hypersensitivity; Richter's Syndrome; Anemia, Hemolytic, Autoimmune; Lymphoma, Mantle-Cell; Drug-Related Side Effects and Adverse Reactions; Pancreatic Neoplasms; Hodgkin Disease; Carcinoma, Transitional Cell; Arthritis, Rheumatoid; Graft vs Host Disease; Neoplasms; Glioblastoma; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Leukemia, Lymphoid; Squamous Cell Carcinoma of Head and Neck; Leukemia, Hairy Cell; Hematologic Neoplasms; Ovarian Neoplasms; Lymphoma, B-Cell Details
Pirtobrutinib LY 3527727; RXC-005; LOXO-305 Approved Redx Pharma Ltd Jaypirca United States Lymphoma, Mantle-Cell Loxo Oncology Inc 2023-01-27 Purpura, Thrombocytopenic, Idiopathic; Lymphoma, B-Cell, Marginal Zone; Lymphoma, B-Cell; Hematologic Neoplasms; Leukemia; Leukemia, Lymphoid; Renal Insufficiency; Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis; Multiple Myeloma; Lymphoma, Mantle-Cell; Leukemia, B-Cell; Hepatic Insufficiency; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Tirabrutinib hydrochloride GS-4059; ONO-4059 Approved Ono Pharmaceutical Co Ltd ベレキシブル, Velexbru Japan Lymphoma Ono Pharmaceutical Co Ltd 2020-03-25 Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Sjogren's Syndrome; Chronic Urticaria; Arthritis, Rheumatoid; Lymphoma; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell; Pemphigus Details
Zanubrutinib BGB-3111 Approved BeOne Medicines Ltd Brukinsa, 百悦泽 United States Lymphoma, Mantle-Cell Beigene (Usa) Inc 2019-11-14 Lymphoma, Follicular; Carcinoma, Non-Small-Cell Lung; Melanoma; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphohistiocytosis, Hemophagocytic; Lymphoma, T-Cell; Lymphoma; Waldenstrom Macroglobulinemia; Hepatic Insufficiency; Leukemia, B-Cell; Anemia, Hemolytic, Autoimmune; Primary mediastinal B cell lymphoma; Lymphoma, Mantle-Cell; Lymphoma, B-Cell; Lung Diseases; Glomerulonephritis, Membranous; Lupus Nephritis; Neoplasms; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Immunoglobulin G4-Related Disease; Nephrosis; Leukemia; Solid tumours; Lymphoma, B-Cell, Marginal Zone Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Nemtabrutinib ARQ-531; MK-1026 Phase 3 Clinical Arqule Inc Hematologic Neoplasms; Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Richter's Syndrome; Hepatic Insufficiency; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Fenebrutinib G-0853; RG-7845; GDC-0853; RO-7010939 Phase 3 Clinical Genentech Inc Arthritis, Rheumatoid; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Lupus Erythematosus, Systemic; Urticaria; Leukemia, Lymphocytic, Chronic, B-Cell Details
Remibrutinib LOU-064; LOU064-NXA; NVP-LOU064-NXA Phase 3 Clinical Novartis Pharma Ag Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Chronic Urticaria; Sjogren's Syndrome; Multiple Sclerosis; Dermatitis; Urticaria; Asthma; Hepatic Insufficiency; Sjogren-Larsson Syndrome; Peanut Hypersensitivity; Hidradenitis Suppurativa; Disease Susceptibility Details
Larotinib Mesylate Z-650 Phase 3 Clinical Guangdong Dongyangguang Pharmaceutical Co Ltd Solid tumours; Esophageal Neoplasms; Pancreatic Neoplasms; Esophageal Squamous Cell Carcinoma Details
Tolebrutinib PRN-2246; SAR-442168 Phase 3 Clinical Principia Biopharma Inc Myasthenia Gravis; Renal Insufficiency; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis; Hepatic Insufficiency Details
Abivertinib A-610MA; AC-0010; AC-0100; AC-001; AC-0010MA; AC-0100-Maleate; EX-ACEA0010MA Phase 3 Clinical Zhejiang Acea Pharmaceutical Co Ltd, Hangzhou Acea Pharmaceutical Research Co Ltd Lymphoma, B-Cell; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Prostatic Neoplasms; Lymphoma, Mantle-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Carcinoma, Non-Small-Cell Lung; Leukemia, Lymphocytic, Chronic, B-Cell Details
Atuzabrutinib PRN-473; SAR-444727 Phase 2 Clinical Principia Biopharma Inc, Sanofi Dermatitis, Atopic Details
Elsubrutinib/Upadacitinib ABBV-599 Phase 2 Clinical Abbvie Inc Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
Poseltinib HM-71224; LY3337641; NB-02 Phase 2 Clinical Hanmi Pharmaceutical Co Ltd Arthritis, Rheumatoid; Lymphoma, Large B-Cell, Diffuse; Central Nervous System Lymphoma; Primary vitreoretinal lymphoma Details
TAS-5315 TAS-5315 Phase 2 Clinical Taiho Pharmaceutical Co Ltd Chronic Urticaria; Arthritis, Rheumatoid Details
HZ-A-018 HZ-A-018 Phase 2 Clinical Hangzhou Yuzheng Pharmaceutical Technology Co Ltd, HeaZen Therapeutics Co Ltd Lymphoma, B-Cell; Multiple Sclerosis; Neuromyelitis Optica; Thrombocytopenia; Central Nervous System Lymphoma Details
Branebrutinib BMS-986195 Phase 2 Clinical Bristol-Myers Squibb Company Arthritis, Rheumatoid; Sjogren's Syndrome; Immune System Diseases; Lupus Erythematosus, Systemic; Dermatitis, Atopic Details
BIIB-091 BIIB-091 Phase 2 Clinical Biogen Inc Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis Details
WXFL10230486 WXFL-10230486; WX-486; HWH-486 Phase 2 Clinical Wuxi Apptec Co Ltd, Humanwell Healthcare (Group) Co Ltd Chronic Urticaria; Arthritis, Rheumatoid Details
M-7583 M7583; M-7583 Phase 2 Clinical Merck & Co Inc Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell Details
Edralbrutinib TG-1701; SHR-1459 Phase 2 Clinical Jiangsu Hengrui Medicine Co Ltd, Jiangsu shengdi Medicine Co Ltd Lymphoma, B-Cell; Nephrosis; Arthritis, Rheumatoid; Autoimmune Diseases; Glomerulonephritis, Membranous; Neuromyelitis Optica; Lymphoma; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
TL-925 TL-925 Phase 2 Clinical Telios Pharmaceuticals Dry Eye Syndromes; Conjunctivitis, Allergic Details
HBW-3210 HBW-3210; HBW3210 Phase 2 Clinical Chengdu Haibowei Pharmaceutical Co Ltd Lymphoma, B-Cell Details
TQB-3702 TQB3702; TQB-3702 Phase 2 Clinical Jiangsu Chia Tai-Tianqing Pharmaceutical Co Ltd Lymphoma, B-Cell; Hematologic Neoplasms; Neoplasms; Chronic Urticaria; Lupus Erythematosus, Systemic Details
HBW-3220 HBW-3220; HBW-3-10; HBW-003 Phase 2 Clinical Chengdu Haibowei Pharmaceutical Co Ltd Lymphoma, B-Cell; Autoimmune Diseases; Lymphoma, Non-Hodgkin; Glomerulonephritis Details
DZD-8586 DZD-8586 Phase 2 Clinical Dizal (Jiangsu) Pharmaceutical Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
BGB-16673 BGB-16673; [14C]-BGB-16673 Phase 2 Clinical BeOne Medicines Ltd Lymphoma, B-Cell, Marginal Zone; Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Neoplasms; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Leukemia, B-Cell; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
HMPL-760 HMPL-760; HMPL760 Phase 2 Clinical Hutchison Medipharma Ltd Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Richter's Syndrome; Lymphoma, Follicular; Lymphoma; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
Rocbrutinib LP-168; NWP-775 Phase 2 Clinical Newave Pharmaceutical Inc Lymphoma, B-Cell, Marginal Zone; Hematologic Neoplasms; Lymphoma, B-Cell; Leukemia, Hairy Cell; Neoplasms; Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis; Neuromyelitis Optica; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
MH-048 MH-048; MH048 Phase 2 Clinical Minghui Pharmaceutical (Shanghai) Co Ltd Lymphoma, B-Cell Details
Elsubrutinib ABBV-105 Phase 2 Clinical Abbvie Ltd Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
CX-1440 CX1440; CX-1440 Phase 2 Clinical Hangzhou Sanyintai Pharmaceutical Technology Co Ltd, Hangzhou Aojin Biomedical Technology Co Ltd Lymphoma, B-Cell; Purpura, Thrombocytopenic, Idiopathic; Graft vs Host Disease; Multiple Sclerosis; Lupus Erythematosus, Systemic; Urticaria; Leukemia, B-Cell; Thrombocytopenia Details
JNJ-64264681 JNJ-4681; JNJ-64264681 Phase 1 Clinical Johnson & Johnson Solid tumours; Hematologic Neoplasms; Neoplasms; Myelodysplastic Syndromes; Prostatic Neoplasms, Castration-Resistant; Lymphoma, Non-Hodgkin; Leukemia, Myeloid, Acute; Leukemia, Lymphocytic, Chronic, B-Cell Details
PCI-45292 Phase 1 Clinical Pharmacyclics Llc Arthritis, Rheumatoid; Autoimmune Diseases Details
BMS-935177 Phase 1 Clinical Bristol-Myers Squibb Company Immune System Diseases Details
BT-1053 BT-1053 Phase 1 Clinical Chengdu Brilliant Pharmaceutical Co Ltd, ScinnoHub Pharmaceutical Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
BTK-Max BTK-Max Phase 1 Clinical Bristol-Myers Squibb Company Arthritis, Rheumatoid; Psoriasis Details
DTRMWXHS-12 DTRMWXHS-12; DTRM-12 Phase 1 Clinical Zhejiang Dtrm Biopharma Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
FCN-647 FCN-647 Phase 1 Clinical Fochon Pharmaceuticals Ltd Lymphoma, B-Cell; Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
SN-1011 SN-1011 Phase 1 Clinical Sinomab Bioscience Ltd Lupus Erythematosus, Systemic Details
AC-0058TA AC-0058; AC-0058TA Phase 1 Clinical Hangzhou Acea Pharmaceutical Research Co Ltd, Zhejiang Acea Pharmaceutical Co Ltd Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
BI-BTK-1 BI-BTK-1 Phase 1 Clinical C.H. Boehringer Sohn Ag & Co. Kg Lupus Nephritis Details
DTRM-505 DTRM-505 Phase 1 Clinical Lymphoma, B-Cell; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
DWP-212525 DWP-212525 Phase 1 Clinical Daewoong Pharmaceutical Co Ltd Autoimmune Diseases; Arthritis, Rheumatoid; Lupus Erythematosus, Systemic; Pemphigus Details
DWP-213388 DWP-213388 Phase 1 Clinical Daewoong Pharmaceutical Co Ltd Autoimmune Diseases Details
NX-5948 NX-5948 Phase 1 Clinical Nurix Therapeutics Inc Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
UBX-303061 UBX-303061 Phase 1 Clinical Ubix Therapeutics Inc Lymphoma, B-Cell Details
[14C]Pirtobrutinib LOXO-305; [14C]RXC-005; RXC-005; [14C]LOXO-305 Phase 1 Clinical Redx Pharma Ltd Details
ANG-0623 ANG-0623; ANG0623 Phase 1 Clinical Angel Pharmaceuticals Co Ltd Multiple Sclerosis Details
XS-04 XS-04 Phase 1 Clinical Jiangsu Xingsheng Xinhui Pharmaceutical Co Ltd Hematologic Neoplasms; Lymphoma, Large B-Cell, Diffuse Details
HZ-Q1070 HZ-Q1070; HZ-Q-1070 Phase 1 Clinical HeaZen Therapeutics Co Ltd Lymphoma, B-Cell; Neoplasms Details
ABBV-101 ABBV-101 Phase 1 Clinical Abbvie Inc Hematologic Neoplasms Details
IMG-004 IMG-004 Phase 1 Clinical Hutchmed (China) Ltd Chronic Urticaria Details
XNW-1011 EVER001; EVER-001; XNW1011; XNW-1011; SN-1011; SN1011 Phase 1 Clinical Suzhou Sinovent Pharmaceuticals Co Ltd, Sinomab Bioscience Ltd Lymphoma, B-Cell; Autoimmune Diseases; Glomerulonephritis, Membranous; Multiple Sclerosis; Neuromyelitis Optica; Lupus Erythematosus, Systemic; Nephrotic Syndrome; Pemphigus Details
AC-0676 AC0676; AC-676; AC676; AC-0676 Phase 1 Clinical Accutar Biotechnology Inc Hematologic Neoplasms; Lymphoma, B-Cell; Autoimmune Diseases Details
JDB175 JDB175 Phase 1 Clinical Shanghai Jiabao Yaoyin Pharmaceutical Technology Co Ltd Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis Details
SS-001 SS-001 Phase 1 Clinical Zibo Baijichangsheng Pharmaceutical Co Ltd Lymphoma, B-Cell Details
BMS-986196 11C-BMS-986196 Phase 1 Clinical Bristol-Myers Squibb Company Multiple Sclerosis Details
Docirbrutinib AS-1763; BN-102; CB-1763 Phase 1 Clinical Bionova Pharmaceuticals (Shanghai) Ltd, Carna Biosciences Inc Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Leukemia, B-Cell; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Sofnobrutinib AS-0871; AS-871 Phase 1 Clinical Carna Biosciences Inc Autoimmune Diseases Details
NX-2127 NX-2127 Phase 1 Clinical Nurix Therapeutics Inc Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell; Central Nervous System Lymphoma Details
TT-01488 TT-01488 Phase 1 Clinical TransThera Sciences (Nanjing) Inc Lymphoma, B-Cell; Solid tumours; Leukemia, B-Cell Details
SYHA-1811 SYHA-1811 Phase 1 Clinical Shanghai Runshi Pharmaceutical Technology Co Ltd Lymphoma, B-Cell Details
HSK-29116 HSK-29116 Phase 1 Clinical Sichuan Haisco Pharmaceutical Co Ltd Lymphoma, B-Cell Details
YZJ-3058 Phase 1 Clinical Shanghai Haiyan Pharmaceutical Technology Co Ltd Arthritis, Rheumatoid; Lymphoma, Large B-Cell, Diffuse; Leukemia, Lymphocytic, Chronic, B-Cell Details
ZXBT-1158 ZXBT-1158 Phase 1 Clinical Guangzhou BeBetter Medicine Technology Co Lymphoma, B-Cell; Multiple Sclerosis Details
Luxeptinib CG026806; CG-806; CG’806; CG-026806 Phase 1 Clinical Crystalgenomics Inc Hematologic Neoplasms; Myelodysplastic Syndromes; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Leukemia, Myeloid, Acute; Leukemia, Lymphocytic, Chronic, B-Cell Details
Evobrutinib M-2951; MSC-2364447; MSC-2364447-C; MSC2364447C Phase 1 Clinical Merck Serono Multiple Sclerosis, Relapsing-Remitting; Renal Insufficiency; Arthritis, Rheumatoid; Multiple Sclerosis; Lupus Erythematosus, Systemic; Hepatic Insufficiency Details
GB-5121 GB-5121; GB5121 Clinical Gossamer Bio Inc Neurolymphomatosis; Central Nervous System Lymphoma Details

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