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Your Position: Home > CNR1

CNR1

Brief Information

Name:Cannabinoid CB1 receptor
Target Synonym:Cannabinoid Receptor 1 (Brain),CNR1,Cannabinoid Receptor 1,CANN6,CB-R,CNR,CB1,Central Cannabinoid Receptor,CB1K5,CB1A,CB1R,Receptor, Cannabinoid, CB1
Number of Launched Drugs:2
Number of Drugs in Clinical Trials:30
Lastest Research Phase:Phase 3 Clinical

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By Product Status:
By Product Category:
By Species:
By Conjugate:
Cat. No. Species Product Description Structure Purity Feature
CN1-H55D3 Human Human CNR1 Protein, Flag,His Tag (Detergent)
CN1-H55D3-structure
CN1-H55D3-sds
CN1-H52P6 Human Human CNR1 Full Length Protein (VLP)
ACRO Quality

Part of Bioactivity data

CN1-H55D3-SPR
 CNR1 SPR

Anti-CNR1 Antibody, Human IgG4 captured on Protein A Chip can bind Human CNR1 Protein, Flag,His Tag (Cat. No. CN1-H55D3) with an affinity constant of 42.8 nM as determined in a SPR assay (in presence of LMNG and CHS) (Biacore 8K) (Routinely tested).

CN1-H52P6-ELISA
 CNR1 ELISA

Immobilized Human CNR1 Full Length Protein-VLP (Cat. No. CN1-H52P6) at 5 μg/mL (100 μL/well) can bind Human Anti-CNR1,Human IgG4 | Human Kappa with a linear range of 1-31 ng/mL (QC tested).

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Cannabidiol/Dronabinol THC-5; delta-9-THC/CBD; MPL-001; MPL-005; GW-1000; KL16-012; BOL-DP-o-04; GW-1000-02; PPP-001; MGC-ODT Approved Gw Pharmaceuticals Sativex, Qixleef Canada Muscle Spasticity; Neuralgia; Cancer Pain; Chronic Pain; Multiple Sclerosis null 2005-04-01 Dementia; Panic Disorder; Phobia, Social; Neuralgia, Postherpetic; Huntington Disease; Reflex Sympathetic Dystrophy; Tourette Syndrome; Muscle Spasticity; Malnutrition; Sciatica; Acute Pain; Neuromyelitis Optica; Arthritis, Psoriatic; Neuralgia; Urinary Bladder, Overactive; Back Pain; Osteoarthritis, Knee; Hepatic Insufficiency; Stress Disorders, Post-Traumatic; Healthy Aging; Hidradenitis Suppurativa; Agoraphobia; Drug Resistant Epilepsy; Renal Insufficiency, Chronic; Social Behavior; Corticobasal degeneration; Cerebral Palsy; Low Back Pain; Agitation; Sleep Initiation and Maintenance Disorders; Peripheral Nervous System Diseases; Genital Diseases, Male; Pain; Chronic Pain; Depression; Depressive Disorder, Major; Marijuana Abuse; Marijuana Use; Spasm; Squamous Cell Carcinoma of Head and Neck; Cancer Pain; Renal Insufficiency; Migraine Disorders; Spinal Cord Injuries; Neoplasms; Arthritis, Rheumatoid; Neck Pain; Diabetic Neuropathies; Sleep Wake Disorders; Opioid-Related Disorders; Essential Tremor; Anorexia; Details
Cannabidiol AVCN-583601; GLA-015; BTX-1503; BTX-1801; BTX-1702; LYT-310; RAD011; PBX-1308; RAD-011; BRCX-014; RLS-103; GWP-42003; GWP-42003-P; BOL-DP-o-05; GW-42003; BTX-1204; ZYN-002; PTL-101; CHI-902; APH-1501 Approved Gw Pharmaceuticals Plc Epidiolex, Epidyolex, Zygel, Cannepil United States Epilepsies, Myoclonic; Lennox Gastaut Syndrome null 2018-06-25 Tobacco Smoking; Migraine Disorders; Peripheral Nervous System Diseases; Acne Vulgaris; HIV Infections; Ovarian Neoplasms; Sleep Initiation and Maintenance Disorders; Facial Pain; Substance-Related Disorders; Marijuana Smoking; Tobacco Use Cessation; Seizures; Tuberous Sclerosis; Pain; Schizophrenia; Chronic Pain; Marijuana Use; Anxiety; Rett Syndrome; Appetitive Behavior; Autism Spectrum Disorder; Marijuana Abuse; Brain Injuries, Traumatic; Depression; Alcoholic Intoxication; Inflammatory Bowel Diseases; Fatty Liver; Child Behavior Disorders; Diabetes Mellitus, Type 2; Spinal Cord Injuries; Muscle injury; Neoplasms; Psychotic Disorders; Opioid-Related Disorders; Diabetic Neuropathies; Coronavirus Disease 2019 (COVID-19); Musculoskeletal Pain; Anxiety Disorders; Sleep Wake Disorders; Graft vs Host Disease; Blepharospasm; Dyspepsia; Arthritis, Rheumatoid; Hyperalgesia; Chronic Urticaria; Hoarding Disorder; Bipolar Disorder; Pancreatic Neoplasms; Brain Diseases; Dysmenorrhea; Sturge-Weber Syndrome; Memory; Mult Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Dronabinol(AXIM Biotechnologies) Phase 3 Clinical Axim Biotechnologies Inc Neoplasms; Nutrition Disorders; Child Nutrition Disorders; Vomiting; Nausea; Cachexia; Sarcopenia; Anorexia Nervosa Details
Adezunap AP-707 Phase 3 Clinical CannaXan GmbH Stroke; Peripheral Nerve Injuries; Diabetes Mellitus; Low Back Pain; Accidental Injuries; Diabetic peripheral neuropathy; Neuralgia; Back Pain; Phantom Limb; Multiple Sclerosis; Peripheral Nervous System Diseases; Brachial Plexus Neuropathies; Somatoform Disorders; Diabetic Neuropathies; Pain, Postoperative; Paraplegia; Chronic Pain; Brain Injuries, Traumatic; Pain Details
Dronabinol(Vertanical) VER-01 Phase 3 Clinical Vertanical GmbH Low Back Pain Details
cannabidiol (Cardiol Therapeutics) Phase 3 Clinical Cardiol Therapeutics Inc Coronavirus Disease 2019 (COVID-19); Pericarditis; Cardiovascular Diseases; Myocarditis Details
V-24343 V-24343; ANEB-001 Phase 2 Clinical Vernalis Plc Poisoning; Obesity Details
11C-MePPEP 11C-MePPEP Phase 2 Clinical Eli Lilly And Company Substance-Related Disorders; Obesity Details
AX-1602 AX-1602 Phase 2 Clinical Axim Biotechnologies Inc Psoriasis; Dermatitis, Atopic; Vitiligo Details
Nimacimab RYI-018; RYI-028; JNJ-2463 Phase 2 Clinical Bird Rock Bio Inc Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Renal Insufficiency, Chronic; Diabetic Gastroparesis Details
ART-2713 NEO-1940; ART-2713; ART27.13; AZD-1940 Phase 2 Clinical Astrazeneca Plc, Neomed Inc, Pfizer Inc Weight Loss; Pain; Anorexia; Cachexia; Low Back Pain Details
AEF-0217 AEF-0217 Phase 2 Clinical Aelis Farma Down Syndrome Details
Monlunabant S-MRI-1891; (-)-MRI-1891; NN9440–INV-202; INV-202; MRI-1891 Phase 2 Clinical Inversago Pharma Inc Metabolic Syndrome; Metabolic Diseases; Diabetic Nephropathies; Obesity Details
C20T5 C20T5 Phase 2 Clinical Murdoch Childrens Research Institute Details
C12T12 C12T12 Phase 2 Clinical Murdoch Childrens Research Institute Details
Tetrahydrocannabinol valine hemisuccinate (Skye Bioscience) NB-1111; Sb-100 OE; SBI-100 OE; THC-VHS-NEC; THCVHS; SBI-100; THCVHS-N; UM-5050; THCVHS-NE Phase 2 Clinical University Of Mississippi Glaucoma, Open-Angle; Glaucoma; Ocular Hypertension Details
IGC-AD1 IGC-AD1 Phase 2 Clinical University Of South Florida Dementia; Psychomotor Agitation; Alzheimer Disease Details
AEF-0117 AEF-0117 Phase 2 Clinical National Institute On Drug Abuse, Aelis Farma Marijuana Abuse Details
[11C]OMAR [11C]JHU-75528 Phase 1 Clinical Johns Hopkins University School Of Medicine Schizophrenia; Marijuana Abuse Details
ZYN-001 ZYN-001 Phase 1 Clinical Zynerba Pharmaceuticals Neuralgia; Fibromyalgia Details
Tetrahydrocannabivarin GWP-42004; THCV; O-4394; DELTA9-THCV; GW-42004 Phase 1 Clinical Gw Pharmaceuticals Plc Diabetes Mellitus, Type 2; Metabolic Syndrome; Obesity, Morbid; Hypercholesterolemia; Hyperglycemia; Dyslipidemias Details
Cannabidiol/hydroxychloroquine IHL-675A; IHL-675 Phase 1 Clinical Incannex Healthcare Ltd Arthritis, Rheumatoid; Respiratory Distress Syndrome, Adult Details
Zevaquenabant MRI-1867; (S)-MRI-1867; INV-101 Phase 1 Clinical National Institutes Of Health Scleroderma, Systemic Details
Atorvastatin Calcium Hydrate/Cannabidiol Phase 1 Clinical Indication Bioscience LLC Coronary Disease; Dyslipidemias Details
TPT0301 TPT-0301; TPT0301 Phase 1 Clinical Tetra Pharm Technologies ApS Chronic Pain Details
INV-347 NN9441; NN-9441; INV-347 Phase 1 Clinical Inversago Pharma Inc Obesity Details
IPI 201(Isosceles Pharmaceuticals Inc ) IPI-201 Phase 1 Clinical Pain, Postoperative Details
GFB-024 Phase 1 Clinical Takeda Pharma Kidney Diseases; Endocrine System Diseases; Diabetes Complications; Diabetic Nephropathies; Diabetes Mellitus Details
DBPR-211 Phase 1 Clinical National Health Research Institutes Diabetes Mellitus, Type 2 Details
MP-10X MP-10X Clinical Medipure Holdings Pain Details
MP-20X MP-20X Clinical Medipure Holdings Mood Disorders; Anxiety Disorders Details
Cannabidiol (Receptor Life Sciences) Clinical Receptor Life Sciences Inc Autism Spectrum Disorder Details
Cannabidiol/Palmitoylethanolamide THX-210; SCI–210 Clinical Therapix Biosciences Ltd Autism Spectrum Disorder; Diabetic Neuropathies Details

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