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DRD1

Brief Information

Name:Dopamine D1 receptor
Target Synonym:D(1A) dopamine receptor,DRD1,Dopamine Receptor D1,Dopamine D1 Receptor,DRD1A,DADR,Receptors, Dopamine D1
Number of Launched Drugs:8
Number of Drugs in Clinical Trials:16
Lastest Research Phase:Approved

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Cat. No. Species Product Description Structure Purity Feature
DR1-H52P6 Human Human DRD1 Full Length Protein (VLP)
ACRO Quality

Public Drug Information

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Docarpamine TA-870; TA-8704 Approved Tanadopa Heart Failure null 1994-01-01 Heart Failure Details
Olanzapine/Fluoxetine hydrochloride OFC Approved Eli Lilly And Company Symbyax United States Bipolar Disorder Eli Lilly And Company 2003-12-24 Depressive Disorder, Major; Bipolar Disorder; Depressive Disorder; Depressive Disorder, Treatment-Resistant Details
Zuclopenthixol Hydrochloride LU-0108 Approved Clopixol Bipolar Disorder; Schizophrenia null 1962-01-01 Schizophrenia; Bipolar Disorder Details
Methylergometrine Maleate Approved Metenarin, Methergine, Ryegonivin, Basofortina, Methylergobrevin Postpartum Hemorrhage; Uterine Cervical Incompetence; Uterine Hemorrhage; Uterine Inertia Details
Samidorphan/Olanzapine ALKS-3831 Approved Alkermes Plc Lybalvi United States Bipolar Disorder; Schizophrenia Alkermes Inc 2021-05-28 Schizophrenia; Bipolar Disorder; Psychotic Disorders; Bipolar and Related Disorders; Bipolar I Disorder; Alcoholism Details
Olanzapine ALKS-7921; LY-170052; LY-170053; INP-105 Approved Eli Lilly And Company Lanzac, Midax, Zypadhera, Zalasta, Zyprexa, Zyprexa Velotab, Zyprexa Relprevv, Olansek, Zyprexa Zydis, Olanzapine ODF, 再普乐 EU Schizophrenia; Bipolar Disorder null 1996-09-27 Emergence Delirium; Anorexia Nervosa; Fasting; Chemotherapy-induced nausea and vomiting; Cachexia; Borderline Personality Disorder; Bipolar II Disorder; Depressive Disorder, Treatment-Resistant; Nausea; Gambling; Vomiting; Autistic Disorder; Bipolar I Disorder; Feeding and Eating Disorders; Postoperative Nausea and Vomiting; Multiple Myeloma; Weight Loss; Malaria, Falciparum; Insulin Resistance; Bipolar Disorder; Anorexia; Opioid-Related Disorders; Neoplasms; Stomach Neoplasms; Depression; Esophageal Neoplasms; Depressive Disorder, Major; Schizophrenia; Biliary Tract Neoplasms; Solid tumours; Hematopoietic stem cell transplantation (HSCT); Substance-Related Disorders Details
Phenylpropanolamine Hydrochloride Approved Nasadec, Nasathera, Pararhinol Nasal Obstruction Details
Olanzapine/Hydroxyzine pamoate Approved Nausea Details
Stepholidine Approved Mainland China Attention Deficit Disorder with Hyperactivity; Tourette Syndrome; Migraine Disorders; Headache null 1995-01-01 Migraine Disorders; Headache; Attention Deficit Disorder with Hyperactivity; Tourette Syndrome Details

Clinical Drug Information

Name Research Code Research Phase Company Indications Clinical Trials
Ecopipam PSYRX-101; Sch-39166 Phase 3 Clinical Merck Sharp & Dohme Corp Language Disorders; Speech Disorders; Self-Injurious Behavior; Lesch-Nyhan Syndrome; Childhood-Onset Fluency Disorder; Tourette Syndrome; Gambling; Stuttering Details
Tavapadon CVL-751; PF-6649751; PF-06649751 Phase 3 Clinical Pfizer Inc, Cerevel Therapeutics Llc Renal Insufficiency; Parkinson Disease; Hepatic Insufficiency Details
Thioridazine TP-21 Phase 3 Clinical Novartis Pharma Ag Schizophrenia; Anxiety Disorders; Carcinoma, Hepatocellular Details
Olanzapine long acting injectable (Teva Pharmaceutical Industries) TV-44749; TEV-‘749; mdc-TJK; TEV-749 Phase 3 Clinical Medincell SA Schizophrenia Details
Olanzapine/samidorphan (Qilu Pharmaceutical) Phase 3 Clinical Qilu Pharmaceutical Co Ltd Schizophrenia Details
PF-06412562 PF-6412562; PF-06412562 Phase 2 Clinical Pfizer Inc Schizophrenia; Schizophrenia Spectrum and Other Psychotic Disorders; Parkinson Disease Details
Mevidalen LY-3154207 Phase 2 Clinical Eli Lilly And Company Alzheimer Disease; Parkinson Disease; Lewy Body Disease Details
TGOF02N TGOF-02N; TGOF02N; FKF02SC Phase 2 Clinical Fabre-Kramer Schizophrenia Details
Docarpamine (Martin Pharmaceuticals) Phase 2 Clinical Martin Pharmaceuticals Inc Gastrointestinal Diseases; Liver Cirrhosis; Mouth Diseases Details
Razpipadon CVL-871 Phase 2 Clinical Pfizer Inc Dementia Details
UCB-0022 UCB-0022 Phase 2 Clinical Ucb Biopharma Srl Parkinson Disease Details
[11C]NNC-112 [11C]NNC-112 Phase 2 Clinical Glaxosmithkline Plc Diagnostic agents Details
Lu-AF-28996 Phase 1 Clinical H. Lundbeck A/S Parkinson Disease Details
asenapine schizophrenia (Livzon Pharmaceutical/LTS Lohmann Therapie-Systeme) Phase 1 Clinical Lts Lohmann Therapie-Systeme Ag Schizophrenia Details
Olanzapine intranasal (Neurelis) NRL-4; NRL-1004 Phase 1 Clinical Neurelis Inc Bipolar Disorder Details
Oxytocin/Methylergometrine Maleate Phase 1 Clinical Nanjing Gritpharma Co Ltd Hemorrhage; Obstetric Labor Complications Details
ITI-333 ITI-333 Phase 1 Clinical Intra-Cellular Therapies Inc Pain; Mood Disorders; Opioid-Related Disorders Details
PF-06730110 PF-06730110; [18F]MNI-968 Phase 1 Clinical Invicro Llc Nerve Degeneration Details

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